1. Junwei Wang#, Quanjin Rong#, Lei Ye#, Bingqian Fang#, Yifan Zhao,Yu Sun, Haikun Zhou, Dan Wang, Jinting He, Zhenzhen Cui, Qijian Zhang, Di Kang*, Lihong Hu*. Discovery of a Novel Orally Bioavailable FLT3-PROTAC Degrader for Efficient Treatment of Acute Myeloid Leukemia and Overcoming Resistance of FLT3 Inhibitors, Journal of Medicinal Chemistry. 2024, 67(9):7197-7223(共同通讯,中科院一区,IF=4.7).
2. Lei Ye#, Zhenzhen Cui#, Yu Sun#, Haikun Zhou, Quanjin Rong, Dan Wang, Jiaming Jin, Qijian Zhang, Di Kang*, Lihong Hu*, Junwei Wang*. Discovery of a potent Gilteritinib-based FLT3-PROTAC degrader for the treatment of Acute myeloid leukemia, Bioorganic Chemistry. 2024, Aug:149:107477(共同通讯,中科院一区,IF=4.7).
3. Jiaming Jin#, Zhenzhen Cui#, Cheng Lv#, Xuemei Peng, Zhiqi Yan, Yi Song, Yu Cao, Wenyi Zhou, Enpeng Wang, Xufan Chen, Di Kang*, Lihong Hu*, Junwei Wang*. Design, synthesis, and biological evaluation of a series of indolone derivatives as novel FLT3 inhibitors for the treatment of acute myeloid leukemia. Bioorganic Chemistry, 2023, 138:106645(共同通讯,中科院一区,IF=4.7).
4. Di Kang#*, Yan Liu#, Yi Song#, Bingqian Fang, Qichun Zhang, Lihong Hu*. Triptolide Shows High Sensitivity and Low Toxicity Against Acute Myeloid Leukemia Cell Lines Through Inhibiting WSTF-RNAPII Complex, Frontiers in oncology. 2022, 12(811850) (共一/共同通讯,中科院三区,IF=3.3).
5. Di Kang#, Xiang Pan#, Yi Song#, Yan Liu, Dan Wang, Xuejun Zhu, Junwei Wang*, Lihong Hu*. Discovery of a novel water-soluble, rapid-release triptolide prodrug with improved drug-like properties and high efficacy in human acute myeloid leukemia. European Journal of Medicinal Chemistry, 2022, 243(114694) (共一,中科院一区,IF=5.9).
6.Junwei Wang#*, Xiang Pan#, Yi Song#, Jian Liu, Fei Ma, Ping Wang, Yan Liu, Lin Zhao, Kang*, Lihong Hu*. Discovery of a Potent and Selective FLT3 Inhibitor (Z) N (5-((5-Fluoro-2-oxoindolin-3-ylidene)methyl)-4-methyl 1H pyrrol-3-yl)-3-(pyrrolidin-1-yl)propenamide with Improved Drug-like Properties and Superior Efficacy in FLT3-ITD-Positive Acute Myeloid Leukemia. Journal of Medicinal Chemistry, 2021, 64(8): 4870-4890(共同通讯,中科院一区,IF=6.8).